Effects of penfluridol on dopamine-sensitive adenylate cyclase in corpus striatum and substantia nigra of rats |
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Authors: | U. Seeber K. Kuschinsky |
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Affiliation: | (1) Abteilung Biochemische Pharmakologie, Max-Planck-Institut für Experimentelle Medizin, Hermann-Rein-Strasse 3, D-34 Göttingen, Germany |
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Abstract: | Summary Penfluridol, a neuroleptic with diphenylbutyl piperidine structure, blocked the dopamine-sensitive adenylate cyclase in homogenates of corpus striatum and substantia nigra of rats, probably by a competitive antagonism versus dopamine.Acknowledgment. We thank Dr P. Janssen (Beerse, Belgium) for a generous gift of penfluridol. |
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