| 钯催化的吲哚嗪与苯硼酸氧化偶联反应 |
| |
| 引用本文： | 杨誉竹,沈创,张玉红. 钯催化的吲哚嗪与苯硼酸氧化偶联反应[J]. 中国科技论文在线, 2013, 0(12): 1302-1306,1309 |
| |
| 作者姓名： | 杨誉竹 沈创 张玉红 |
| |
| 作者单位： | 浙江大学化学系,杭州301127 |
| |
| 基金项目： | 高等学校博士学科点专项科研基金资助项目（20110101110006） |
| |
| 摘 要： | 报道了一种钯催化下碳酸银作为氧化剂的吲哚嗪芳基化的新方法。该方法使用易得的苯硼酸，可以高收率地选择性在吲哚嗪的C-3位发生芳基化反应，而且底物适用性广，官能团耐受性好。
|
| 关 键 词： | C—H键活化 吲哚嗪 钯催化 苯硼酸 芳基化 |
Pd-catalyzed oxidative coupling of indolizines with arylboronic acids |
| |
| Yang Yuzhu,Shen Chuang,Zhang Yuhong. Pd-catalyzed oxidative coupling of indolizines with arylboronic acids[J]. Sciencepaper Online, 2013, 0(12): 1302-1306,1309 |
| |
| Authors: | Yang Yuzhu Shen Chuang Zhang Yuhong |
| |
| Affiliation: | (Department of Chemistry, Zhej iang University, Hangzhou , Zhej iang 310027, China) |
| |
| Abstract: | A new method of Pd-catalyzed direct arylation of indolizines with arylboronic acids employing Ag2 CO3 as the oxidant has been established. The approach can provide an efficient access to diverse @3 arylated indolizines with high yields, wide sub- strate scope and excellent functional group tolerance. |
| |
| Keywords: | C--H activation indolizines Pd-catalysis arylboronic acids arylation |
| 本文献已被 维普 等数据库收录！ |
