| 3-(4-氯苯基)-1,3-2H-3-苯基恶唑[3,4-a]吲哚合成 |
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| 引用本文： | 端木慧.3-(4-氯苯基)-1,3-2H-3-苯基恶唑[3,4-a]吲哚合成[J].新乡学院学报(自然科学版),2012(4):319-321. |
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| 作者姓名： | 端木慧 |
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| 作者单位： | 西北有色地质勘查局七一一总队 |
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| 摘 要： | 以溴化亚铜作催化剂,DMF作溶剂,用N-(o-alkynylphenyl)imines亚胺在温和条件下环合-加成反应,一步合成吲哚衍生物,结果发现恶唑类吲哚在不同催化剂、不同底物种类及反应条件下的反应速度和产率具有较大差异性.
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| 关 键 词： | 吲哚 串联反应 恶唑 |
Synthesis of 3-(4-chlorophenyl)-1, 3-2H-3-phenyloxazoleindole |
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| Institution: | DUAN-MU Hui(711 Corps,Northwest Nonferrous Geological Exploration Bureau,Hanzhong 723000,China) |
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| Abstract: | Using cuprous bromide as catalyst,DMF as solvent,indole derivatives are get from N-(o-alkynylphenyl)imines by one step cyclization-addition reaction under mild conditions.Results show that the reaction rate and yield of oxazolidinone indole have great differences under different catalysts,substrate types and reaction conditions. |
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| Keywords: | indole tandem reaction oxazole |
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